Table 3. Pharmacokinetic parameters after single subcutaneous bolus administration of SNF472 into rats.
10 mg/kg | 30 mg/kg | 100 mg/kg | |
---|---|---|---|
Cmax (ng/mL) | 4876 | 61014 | 263264 |
t1/2 (min) | 3.9 | 17.0 | 11.5 |
AUC(0→t) (ng·h/mL) | 1633 | 32646 | 139603 |
MRT (0→∞) (h) | 0.47 | 0.48 | 0.49 |
Vz/F (L/kg) | 0.48 | 0.48 | 0.61 |
Cl/F (L/h/kg) | 0.22 | 0.27 | 0.21 |
Cmax: maximum concentration measured; t1/2: half-life; AUC: area under the curve; MRT: mean residence time; Vz: volume of distribution; Cl: clearance; F: absolute bioavailability