Table 8. Activity of FucC6 and Lea glycopeptide dendrimers against Pseudomonas aeruginosa biofilms.
| Ligand | MBIC a [μM] | MBC b [μM] | Dispersal | MIC c |
| FD2 | 20 | >30 | 100% dispersal at 50 μM | n.i. d |
| FucC6G2 | 9 | >20 | 100% dispersal at 30 μM | >64 μM |
| LeaxG2 | 30 | nd | ∼88% dispersal at 50 μM | nd |
aMBIC is minimal biofilm inhibitory concentration.
bMBC = minimal bactericidal concentration under biofilm forming conditions, determined by CFU counts in the biofilm supernatant.
cMIC = minimal inhibitory concentration in a standard 2-fold dilution assay for antibacterial activity in full LB medium. n.i. = no inhibition in a growth assay using 50 μM compound, nd = not determined.
dFrom ref. 19. See also ESI Fig. S115/S116 (biofilm data), S120 (MIC data), and Table S1 (cell viability data).