Table 5.
IC50 values for monepantel on expressed nAChRs from A. suum and O. dentatum.
IC50 (mean ± s.e.m., n) | |
---|---|
Asu-ACR-16 nAChR | 1.6 ± 3.1 nM; 0.2 ± 2.3 μM, n = 4 |
Ode pyrantel/tribendimidine nAChRs | 1.7 ± 0.7 μM, n = 4 |
Ode levamisole nAChRs | 5.0 ± 0.5 μM, n = 4 |