Table 1.
RGFP966 is an HDAC3 Selective Inhibitor
Inhibitor | Molar mass | Blood–brain barrier permeable? | HDAC1 | HDAC2 | HDAC3 |
---|---|---|---|---|---|
RGFP966 | 362.4 g/mol | Yes | IC50 2.069 μM = 1.97 nmol/g retinal tissue | IC50 3.961 μM = 3.77 nmol/g retinal tissue | IC50 0.064 μM = 0.061 nmol/g retinal tissue |