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. 2018 May 18;8:152. doi: 10.3389/fonc.2018.00152

Table 2.

Clinical trials of drug-conjugated anti-CD33 mAbs other than GO.

Disease type and inclusion criteria Drug or drug combination, other therapies Outcome measures (Estimated) enrollment Clinical trials identifier Trial status
R/R AML
High-risk MDS
CML
Lintuzumab-90Y Primary: toxicity, MTD, and ORR 24 NCT00002890 Completed (2001)

AML, ALL
High-risk MDS
Lintuzumab-90Y + etoposide + aHSCT Primary: MTD, toxicity and engraftment efficacy 24 NCT00006040 Completed (2003)

R/R AML
AML in patients not eligible for curative therapy
ap or bc CML
high-risk MDS
MDS/MPN (CMML)
Lintuzumab-213Bi + cytarabine Primary: MTD 32 NCT00014495 Completed (2009)

R/R AML
ap or bc CML
High-risk MDS
Lintuzumab-225Ac Primary: MTD 23 NCT00672165 Completed (2015)

De novo AML in patients ≥60 years Lintuzumab-225Ac + low-dose cytarabine Primary: MTD
Secondary: toxicity PFS, DFS, and OS
72 NCT02575963 Recruiting (estimated completion early 2019)

Relapsed AML
AML in patients not eligible for curative therapy
Vadastuximab talirine (SGN-CD33A) + AZA or decitabine vs. vadastuximab talirine (SGN-CD33A) monotherapy Primary: AE and LA
Secondary: PK, ADA, CR, DOR, RFS, and OS
195 NCT01902329 Completed late 2017

De novo AML Vadastuximab talirine (SGN-CD33A) during induction with cytarabine and daunorubicin; during consolidation with high-dose cytarabine; as a monotherapy for maintenance Primary: AE, DLT, and LA
Secondary: CR, DFS, OS, PK, ADA, and MRD
116 NCT02326584 Active, not recruiting (estimated completion late 2021)

De novo or secondary AML, intermediate or adverse-risk cytogenetics Vadastuximab talirine (SGN-CD33A) + AZA or decitabine vs. placebo + AZA or decitabine Primary: OS and CR
Secondary: toxicity, MRD level, and EFS
240 NCT02785900 Terminated June 2016 due to higher rate of deaths and infections in verum group

High-risk MDS Vadastuximab talirine (SGN-CD33A) + AZA vs. placebo + AZA Primary: toxicity and ORR
Secondary: toxicity, CR, HI, DOR, PFS, rate of transformation to AML, and OS
19 (142 planned) NCT02706899 Terminated late 2017 due to results from NCT02785900

R/R AML Vadastuximab talirine (SGN-CD33A) + melphalan + fludarabine, followed by aHSCT
Vadastuximab talirine (SGN-CD33A) monotherapy after aHSCT
Primary: AE, 1-year-survival, MRD level
Secondary: DOR and OS
14 NCT02614560 Terminated late 2017 due to results from NCT02785900

R/R AML in patients not eligible for curative therapy Monotherapy with IMGN779 (anti-CD33 mAb indolino benzodiazepine ADC) Primary: MTD
Secondary: AE, ORR, PK, and ADA
124 NCT02674763 Recruiting (estimated completion early 2019)

ADA, anti-drug antibodies; ADC, antibody–drug conjugate; AE, adverse events; aHSCT, allogeneic hematopoietic stem cell transplantation; ALL, acute lymphoblastic leukemia; AML, acute myeloid leukemia; ap, accelerated-phase; AZA, 5-azacytidine; bc, blast-crisis; CML, chronic myeloid leukemia; CMML, chronic myelomonocytic leukemia; CR, complete remission; DFS, disease-free survival; DLT, dose-limiting toxicity; DOR, duration of response; GO, gemtuzumab ozogamicin; HI, hematological improvement; LA, laboratory abnormalities; mAb, monoclonal antibody; MDS, myelodysplastic syndrome; MDS/MPN, myelodysplastic-myeloproliferative neoplasm; MRD, minimal residual disease; MTD, maximum tolerated dose; ORR, overall response rate; OS, overall survival; PFS, progression-free survival; PK, pharmacokinetics; R/R, refractory/relapsed.

Data from http://ClinicalTrials.gov (Accessed: February 20, 2018).