Skip to main content
. 2018 May 4;9(21):4909–4918. doi: 10.1039/c8sc01324a

Table 5. Kinetic resolution of (±)-37.

Inline graphic
Entry Conditions a Conv. (%) 37 er 42 er
1 3 (10 mol%) 55 77 : 23 74 : 26
2 3 (10 mol%) + 14 (1 equiv.) 56 92 : 8 85 : 15
3 3 (10 mol%) + PhCO2H (10 mol%) 53 92 : 8 89 : 11
4 3 (10 mol%) + 48 (10 mol%) 56 92 : 8 83 : 17
5 49 (10 mol%) 64 50 : 50 50 : 50

aSee ESI for reaction times.