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. Author manuscript; available in PMC: 2018 Jul 7.
Published in final edited form as: Eur J Med Chem. 2017 Mar 30;134:185–206. doi: 10.1016/j.ejmech.2017.03.069

Table 5.

Data of in vivo study with U937 xenograft model.

Cpd No. Does
(mg/kg)
Tumor growth inhibition (TGI %) Relative increment ratio (T/C %) Mice body weight (g)
11a 100 51 49 25.04 ± 1.31
MS275 50 60 32 19.77 ± 0.61
Ctrl / / / 25.39 ± 1.18