. 2018 May 14;9(23):5160–5164. doi: 10.1039/c8sc01256c

Table 3. Overcoming the limitation of heterocycles in C–H amination ^a ^, ^b .

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^aReaction conditions: (1) 4a–4g (0.1 mmol), 2a (0.15 mmol), CuOAc (0.15 mmol), K₂HPO₄ (0.1 mmol), DMSO (1 mL), 90 °C, 6 h, N₂. (2) 2 M HCl (2 mL), rt. 20 min.

^bIsolated yield.

^cYields of reactions using 0.3 equiv. of CuOAc are shown in parentheses.

Table 3. Overcoming the limitation of heterocycles in C–H amination a , b .

Table 3. Overcoming the limitation of heterocycles in C–H amination ^a ^, ^b .