Skip to main content
. 2018 May 16;9(6):517–521. doi: 10.1021/acsmedchemlett.8b00126

Table 2. Additional SAR of N,N′-(1,2-Phenylene)dibenzenesulfonamide Derivatives.

graphic file with name ml-2018-00126e_0005.jpg

compd R1 R2 R3 IC50 (μM)
7a m-Cl m-Cl H 5.7
7b m-Cl m-Cl Me 4.3
7c m-Cl, p-Me m-Cl, p-Me H 2.3
7d m-Cl, p-Me m-Cl, p-Me F 3.7