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. Author manuscript; available in PMC: 2019 Jun 19.
Published in final edited form as: Biochemistry. 2018 Mar 28;57(24):3359–3363. doi: 10.1021/acs.biochem.8b00204

Table 1.

Rate Constants for TG2 Oxidation by Cystamine, Cystine, and GSSGa

oxidant kinh/Ki (mM−1 min−1) Ki (mM)
cystineb 0.29 NDd
GSSGb 0.0033 NDd
cystamineb 1.2 >0.6
cystaminec 1.7 >0.1
a

Measured in 50 mM Tris and 1 mM EDTA at pH 7.6 and 22 °C.

b

Determined in a deamidation activity assay.

c

Determined in a transamidation activity assay.

d

Not determined.