Table 1.
Rate Constants for TG2 Oxidation by Cystamine, Cystine, and GSSGa
oxidant | kinh/Ki (mM−1 min−1) | Ki (mM) |
---|---|---|
cystineb | 0.29 | NDd |
GSSGb | 0.0033 | NDd |
cystamineb | 1.2 | >0.6 |
cystaminec | 1.7 | >0.1 |
Measured in 50 mM Tris and 1 mM EDTA at pH 7.6 and 22 °C.
Determined in a deamidation activity assay.
Determined in a transamidation activity assay.
Not determined.