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. 2017 Jul 25;32(1):1012–1028. doi: 10.1080/14756366.2017.1350658

Scheme 5.

Scheme 5.

Reagents and conditions: (a) ROH (6, 9, 11), EDAC, HOBt, DIPEA, anh. DMF, r.t., 2–6 h.