Table 1.

Covalent and non-covalent DprE1inhibitors

Covalent inhibitors			Non covalent inhibitors
Compound	Structure	References	Compound	Structure	References
BTZ043		[23]	1–4 Azaindoles		[34]
DNB1		[35]	2-Carboxyquinoxalines		[32]
377790		[26]	4-AQs		[36]
cBT		[16]	8-Pyrrole-BTZ		[37]
BTO		[38]	1,3-BTZ azide		[39]
VI-9376		[40]	Pyrazolopyridones		[33]
PBTZ		[17]	1,2,4-Triazole containing 1,4-BTZ derivatives		[41]