Table 1.
Synthesized azides 7a–7j.
Entry | Azide | Ar | Yield a |
---|---|---|---|
1 | 7a | Ph | 58 |
2 | 7b | 2-OMe–Ph | 61 |
3 | 7c | 3-OMe–Ph | 97 |
4 | 7d | 4-OMe–Ph | 96 |
5 | 7e | 3-F, 4-OMe–Ph | 96 |
6 | 7f | 4-F–Ph | 41 |
7 | 7g | 3-CF3–Ph | 31 |
8 | 7h | 3-NO2–Ph | 82 |
9 | 7i | 5-1H-indol | 35 |
10 | 7j | 3-furyl | - b |
a Isolated yield; b It was not isolated but was reacted in situ.