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. Author manuscript; available in PMC: 2018 Jun 25.
Published in final edited form as: AIMS Biophys. 2017 Aug 21;4(3):491–527. doi: 10.3934/biophy.2017.3.491

Figure 6.

Figure 6

Superpositions of GPCR represented as thin ribbon structures with ligands as space-filling atoms colored accordingly by antagonists as green, agonists as fuchsia, and negative allosteric modulators as orange. (A) Structures of 29 individual class A GPCR. (B) Structures of 3 class B GPCR. (C) Structures of 4 class C GPCR. (D) Structures of 7 class F GPCR. Class A GPCR: Rho (1F88), ADRB1 (2VT4), ADRB2 (2RH1), H1R (3RZE), D3R (3PBL), 5-HT1B (4IAQ), 5-HT2B (4IB4), M1R (5CXV), M2R (3UON), M3R (4DAJ), M4R (5DSG), A2AR (2YDO), S1P1 (3V2W), LPA1 (4Z34), CB1 (5TGZ), NTSR1 (3ZEV), OX1 (4ZJ8), OX2 (4S0V), CCR4 (3ODU), CCR5 (4MBS), CCR9 (5LWE), NOP (4EA3), κ-OR (4DJH), μ-OR (4DKL), δ-OR (4EJ4), AT1R (4YAY), P2Y1 (4XNW), P2Y12 (4NTJ), PAR1 (3VW7). Class B GPCR: GCGR (5EE7), CRF1R (4K5Y, 4Z9G). Class C GPCR: mGlu1 (4OR2, 5CGC, 5CGD), mGlu5 (4OO9) Class F GPCR: SMO (4JKV, 4N4W, 4OR9, 4QIM, 4QIN, 5L7D, 5L7I).