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. Author manuscript; available in PMC: 2018 Jul 2.
Published in final edited form as: Curr Opin Endocrinol Diabetes Obes. 2017 Feb;24(1):73–79. doi: 10.1097/MED.0000000000000311

Table 1.

List of current SGLT2 inhibitors.

Generic Name Brand Name Available Doses (mg) Administration
canagliflozina Invokana® 100, 300 qam before 1st meal
dapagliflozina Farxiga 5, 10 qam
empagliflozina Jardiance® 10, 25 qam
canagliflozin/metformina Invokamet® 50/500, 50/1000, 150/500, 150/1000 BID with meals, max dose 300mg/2000mg
dapagliflozin/metformina Xigduo XR 5/500, 5/1000, 10/500, 10/1000 qam with food, max dose 10mg/2000mg
empagliflozin/metformina Synjardy® 5/500, 5/1000, 12.5/500, 12.5/1000 BID with meals, max dose 25mg/2000mg
empagliflozin/linagliptina Glyxambi® 10/5, 25/5 qam
Ipragliflozinb Suglat® 25, 50 qam, max dose 100mg
tofogliflozinbc Apleway®, Deberza® 20 qam
luseogliflozinc
remogliflozin etabonatec
ertugliflozinc
sotagliflozinc
a

FDA and EMA approved,

b

Ministry of Health, Labour and Welfare approved in Japan,

c

currently in clinical trials or seeking market approval; qam taken once daily in the morning, BID twice daily