Table 1.
List of current SGLT2 inhibitors.
Generic Name | Brand Name | Available Doses (mg) | Administration |
---|---|---|---|
canagliflozina | Invokana® | 100, 300 | qam before 1st meal |
dapagliflozina | Farxiga™ | 5, 10 | qam |
empagliflozina | Jardiance® | 10, 25 | qam |
canagliflozin/metformina | Invokamet® | 50/500, 50/1000, 150/500, 150/1000 | BID with meals, max dose 300mg/2000mg |
dapagliflozin/metformina | Xigduo™ XR | 5/500, 5/1000, 10/500, 10/1000 | qam with food, max dose 10mg/2000mg |
empagliflozin/metformina | Synjardy® | 5/500, 5/1000, 12.5/500, 12.5/1000 | BID with meals, max dose 25mg/2000mg |
empagliflozin/linagliptina | Glyxambi® | 10/5, 25/5 | qam |
Ipragliflozinb | Suglat® | 25, 50 | qam, max dose 100mg |
tofogliflozinbc | Apleway®, Deberza® | 20 | qam |
luseogliflozinc | |||
remogliflozin etabonatec | |||
ertugliflozinc | |||
sotagliflozinc |
FDA and EMA approved,
Ministry of Health, Labour and Welfare approved in Japan,
currently in clinical trials or seeking market approval; qam taken once daily in the morning, BID twice daily