Table 1.
Single dose inhibition assay against VIM2
| Compound | % Inhibition at 50 μM |
|---|---|
| L-Captopril | 98 |
| Clavulanate | 15 |
| Tazobactam | 25 |
| SAHA | 29 |
| 1 | 12 |
| 2a (zinc salt) | 15 |
| 2b (sodium salt) | 93 |
| 3 | 98 |
| 4 | 18 |
| 5 | 34 |
Single dose inhibition assay against VIM2
| Compound | % Inhibition at 50 μM |
|---|---|
| L-Captopril | 98 |
| Clavulanate | 15 |
| Tazobactam | 25 |
| SAHA | 29 |
| 1 | 12 |
| 2a (zinc salt) | 15 |
| 2b (sodium salt) | 93 |
| 3 | 98 |
| 4 | 18 |
| 5 | 34 |