Table 1. MIC (μg/mL) for Lys2–11 Teixobactin Analogues.
| MIC μg/mL (ATCC strains) | ||||
|---|---|---|---|---|
| Gram
(+) |
Gram
(−) |
|||
| entry | S. aureus | B. subtilis | E. coli | P. aeruginosa |
| Arg10–teixobactin (2)7 | 2 | 0.5 | 64 | NI |
| Lys2 | NIa | NI | NI | NI |
| Lys3 | 4 | 0.25 | 32 | 128 |
| Lys4 | 4 | 1 | 32 | 128 |
| Lys5 | NI | NI | NI | NI |
| Lys6 | NI | NI | NI | NI |
| Lys7 | 32 | 8 | 256 | 256 |
| Lys9b | 6 | 1 | 50 | 100 |
| Lys11 | NI | NI | NI | NI |
| meropenemc | 0.0625 | 0.0625 | 0.03125 | 0.25 |
NI: no inhibition.
The starting concentration is 100 μg/mL.
Used as controls.