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. 2016 Dec 19;1(6):1262–1265. doi: 10.1021/acsomega.6b00354

Table 1. MIC (μg/mL) for Lys2–11 Teixobactin Analogues.

  MIC μg/mL (ATCC strains)
  Gram (+)
Gram (−)
entry S. aureus B. subtilis E. coli P. aeruginosa
Arg10–teixobactin (2)7 2 0.5 64 NI
Lys2 NIa NI NI NI
Lys3 4 0.25 32 128
Lys4 4 1 32 128
Lys5 NI NI NI NI
Lys6 NI NI NI NI
Lys7 32 8 256 256
Lys9b 6 1 50 100
Lys11 NI NI NI NI
meropenemc 0.0625 0.0625 0.03125 0.25
a

NI: no inhibition.

b

The starting concentration is 100 μg/mL.

c

Used as controls.