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. 2017 Apr 20;2(4):1550–1562. doi: 10.1021/acsomega.6b00481

Table 2. HDAC Inhibition Assays (IC50) Using Class I and Class IIa HDAC Isoforms.

  IC50 (μM)
molecule HDAC1 HDAC3/NCOR2 HDAC4 HDAC8
3 0.96 ± 0.6 0.33 ± 0.01 >100 7.02 ± 1.53
13 0.39 ± 0.02 0.35 ± 0.003 >100 1.87 ± 0.42
11b 7.9 ± 0.8 50.2 ± 4.7 >100 >100
11e 5.04 ± 0.07 1.97 ± 0.03 >100 >100
SAHAa 0.123 ± 0.003 0.957 ± 0.07 0.101b 1.52b
trichostatin A (TSA)a       0.624
TMP269a     0.275  
a

Assay-positive controls according to relevant isoform.

b

Data from ref (28).