Table 1. Cancer Cell Line Response to Compound 1 in 7-Day Proliferation Assay (Supporting Information).

cell line	histology	IC50 (μM)	max inhibition (%)
HCC1937	breast	0.030	83
T-42D	breast	0.003	84.0
UACC-812	breast	>2.5	21.0
MX-1 cells	breast	>2.5	36.9
NUGC-3	gastric	0.017	92
KE-97	gastric	0.024	95.7
MV4–11	hematological	0.016	93
Daudi	hematological	0.017	99.3
Karpas-422	hematological	0.085	99.9
HEL 92.1.7	hematological	0.003	91.2
ARH-77	hematological	0.010	97.2
REC-1	hematological	0.022	99.7
IM-9	hematological	0.046	93
KMS-12-BM	hematological	0.006	99
RPMI-8226	hematological	0.009	88.5
OPM-2	hematological	>2.5	22.5
NCI-H2171	lung	0 010	97.7
H-2122	lung	0.027	90
NCI-H1930	lung	>2.5	49.6
NCI-H1651	lung	>2.5	32
A375	skin	0.037	91.1
A2058	skin	0.013	96
GAK	skin	0.016	99.9
Colo829	skin	0.013	51
OVCAR-3	ovarian	0.032	95