Table 2. A and B-Ring SAR in the α-Methyl Series.
Mean of at least two runs.
HS = human serum.
% Activation >179%22.
% Inhibition of net glucose AUC.
Experimentally determined; see Supporting Information.
Mean of at least two runs.
HS = human serum.
% Activation >179%22.
% Inhibition of net glucose AUC.
Experimentally determined; see Supporting Information.