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. 2018 Jun 23;9(7):679–684. doi: 10.1021/acsmedchemlett.8b00145

Table 1. Alkyl Side Chain Modification of the Northern Portion.

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a

OCF3 benzamide was chosen to establish this SAR due to improved rat PK comparing to simple benzamide from initial screening SAR.

b

The data is the mean of at least two determinations.