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. 2018 Jul 5;54(58):8120–8123. doi: 10.1039/c8cc01400k

Table 1. K i values (nM) of OT and peptide analogues for human OTR and vasopressin receptors.

Peptide OTR V1a V1b V2
OTc 1.2 ± 0.3 20 ± 3 >6000 >6000
dOTc 1.6 ± 1.3 388 ± 157 nd >6000
dOToc 1.2 ± 0.9 362 ± 124 nd >6000
dLVTc 3.4 ± 1.0 24 ± 5 nd 4844 ± 1670
dLVToc 6.3 ± 3.6 31 ± 9 nd 5819 ± 1704
AlF-NODA-dLVTc 2.6 ± 1.7 157 ± 26 >6000 >6000
AlF-NODA-dLVToc 3.3 ± 1.5 821 ± 217 nd >6000