Table 3. Calculated inhibition constants for the inhibition of CYP2A13 by NAT, NAB and nicotine.
|
K
i (μM) |
|||
| NNK + NAT | NNK + NAB | NNK + nicotine | |
| OPB | 0.21 | 0.23 | 8.51 |
| HPB | 0.71 | 0.87 | 25.01 |
| OPBA | 0.36 | 0.50 | 6.57 |
|
K
i (μM) |
|||
| NNK + NAT | NNK + NAB | NNK + nicotine | |
| OPB | 0.21 | 0.23 | 8.51 |
| HPB | 0.71 | 0.87 | 25.01 |
| OPBA | 0.36 | 0.50 | 6.57 |