Table 2. In Vitro Inhibition of Cdk-2/A and Cdk-9/T1 by IIIM-290 and Its HCl Salt at 500 nM.
% inhibition (±SD) |
||
---|---|---|
test sample | Cdk-2/A | Cdk-9/T1 |
IIIM-290 | 90 ± 0.2 | 94 ± 0.8 |
IIIM-290·HCl | 85 ± 0.5 | 97 ± 1.2 |
% inhibition (±SD) |
||
---|---|---|
test sample | Cdk-2/A | Cdk-9/T1 |
IIIM-290 | 90 ± 0.2 | 94 ± 0.8 |
IIIM-290·HCl | 85 ± 0.5 | 97 ± 1.2 |