Table 3. Pharmacokinetic Parameters of IIIM-290 and IIIM-290·HCl Salt in BALB/c Mice.
PO, 50 mg/kg |
||
---|---|---|
PK parameter | IIIM-290 | IIIM-290·HCl salt |
T1/2 (h) | 1.92 | 5.06 |
Cmax (ng/mL) | 656 | 1030 |
Tmax (h) | 1.0 | 2.0 |
AUC0–t (ng h/mL) | 2570 | 3600 |
AUC0–∞ | 2570 | 3710 |