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. 2018 Jul 27;3(7):8365–8377. doi: 10.1021/acsomega.8b00801

Table 3. Pharmacokinetic Parameters of IIIM-290 and IIIM-290·HCl Salt in BALB/c Mice.

  PO, 50 mg/kg
PK parameter IIIM-290 IIIM-290·HCl salt
T1/2 (h) 1.92 5.06
Cmax (ng/mL) 656 1030
Tmax (h) 1.0 2.0
AUC0–t (ng h/mL) 2570 3600
AUC0–∞ 2570 3710