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. 2017 May 12;8(7):1421–1434. doi: 10.1039/c7md00105c

Table 2. In vitro inhibition of TNF-α-induced NF-κB activation in the NCI-H460 lung adenocarcinoma cell line.

Compd. IC50 (μM) Compd. IC50 (μM)
2Y1 >20 3Y9 15.51 ± 1.02
2Y2 >20 3Y10 7.13 ± 0.44
2Y4 15.96 ± 0.21 5Y1 14.83 ± 0.38
2Y5 8.04 ± 0.56 5Y2 10.14 ± 0.34
2Y10 10.32 ± 0.29 5Y3 4.80 ± 0.47
2Y11 16.24 ± 0.60 5Y4 3.64 ± 0.52
3Y1 >20 5Y5 2.26 ± 0.48
3Y2 >20 5Y8 0.36 ± 0.08
3Y3 15.17 ± 0.76 5Y9 4.80 ± 0.55
3Y4 >20 5Y10 2.33 ± 0.17
3Y5 5.43 ± 0.68 UA >20
3Y8 0.94 ± 0.27