| NR | Nuclear receptors |
| SAR | Structure-activity relationship |
| PR | Progesterone receptor |
| LXR | Liver X receptor |
| AR | Androgen receptor |
| GR | Glucocorticoid receptor |
| LBD | Ligand-binding domains |
| ROR | retinoic acid receptor-related orphan receptors |
| NPC1 | Niemann-Pick disease type C1 |
| NPC1L1 | Niemann-Pick disease type C1-like 1 |
| OHF | Hydroxyflutamide |
| Ts | p-Toluenesulfonyl |
| EDC | N-Ethyl-N’-(3-dimethylaminopropyl)carbodiimide |
| DMAP | 4-(N,N-Dimethylamino)pyridine |
| DMF | Dimethylformamide |
| SEM | 2-(Trimethylsilyl)ethoxymethyl |
| Cy | Cyclohexyl |
| DMA | Dimethylacetamide |
| TBAF | Tetrabutylammonium fluoride |
| THF | Tetrahydrofuran |