Table 3.
Pharmacokinetic properties of Zl-n-91
| Dosing route |
T1/2 Range(h) |
T1/2 (h) |
Tmax (h) |
Cmax (ng/mL) |
AUC0-t (ng/h/mL) |
AUC0-m (ng/h/mL) |
Vz(F) (L/kg) |
CL(F) (L/h/kg) |
F (%) |
| PO | 4–8 | 1.35 | 2 | 96.5 | 241 | 244 | 39.9 | 20.5 | 33.3 |
| Dosing route |
T1/2 Range(h) |
T1/2 (h) |
C0 | CL | AUC0-t (ng/h/mL) |
AUC0-m (ng/h/mL) |
Vss | MRTinf (h) |
|
| IV | 0.5–4 | 0.62 | 6030 | 6.87 | 725 | 728 | 2.31 | 0.34 | |