Figure 9.
(a) Electrostatic potential map of Pseudomonas GABA-AT active site region. Blue, red and white colors represent regions with positive, negative and neutral electrostatic potential value, respectively; (b) GABA derivatives bound into the Pseudomonas GABA-AT catalytic site; (c) (S)-Pregabalin analogues bound into the Pseudomonas GABA-AT catalytic site; (d) (R)-Pregabalin analogues bound into the Pseudomonas GABA-AT catalytic site; (e) (S)-Baclofen analogues bound into the Pseudomonas GABA-AT catalytic site; (f) (R)-Baclofen analogues bound into the pseudomonas GABA-AT catalytic site. PLP prosthetic group is shown as spacefill model.
