Table 1.
Code | Structure | MbtI Residual Activity at 100 μM | MbtI IC50 (μM) |
---|---|---|---|
I | 11.0 ± 3.9 | 11.6 ± 2.4 | |
1 | 23.3 ± 3.4 | 55.8 ± 4.2 | |
1b | >75 | ND | |
2 | 28.1 ± 2.9 | 61.3 ± 5.3 | |
3 | >75 | ND | |
4 | >75 | ND | |
5 | 50.1 ± 7.1 | ND |
ND: not determined.
Code | Structure | MbtI Residual Activity at 100 μM | MbtI IC50 (μM) |
---|---|---|---|
I | 11.0 ± 3.9 | 11.6 ± 2.4 | |
1 | 23.3 ± 3.4 | 55.8 ± 4.2 | |
1b | >75 | ND | |
2 | 28.1 ± 2.9 | 61.3 ± 5.3 | |
3 | >75 | ND | |
4 | >75 | ND | |
5 | 50.1 ± 7.1 | ND |
ND: not determined.