. 2018 Jul 10;61(15):6830–6845. doi: 10.1021/acs.jmedchem.8b00718

Table 2. Analogs of Hit Compounds 5, 19, and 21 with Their Respective HTR2A, DRD2, and HRH1 Docking Ranks, Binding Constants, and Selectivity Ratios^a.

Footnotes: *Weak binding detected at high concentration but K_i could not be calculated. ^aNo agonist activity measured in calcium flux assay at concentrations up to 100 μM.

Table 2. Analogs of Hit Compounds 5, 19, and 21 with Their Respective HTR2A, DRD2, and HRH1 Docking Ranks, Binding Constants, and Selectivity Ratiosa.

Table 2. Analogs of Hit Compounds 5, 19, and 21 with Their Respective HTR2A, DRD2, and HRH1 Docking Ranks, Binding Constants, and Selectivity Ratios^a.