Supplementary Table 1.
known therapeutic targets of CML.
| ESR1 | MLL | IMD21 | QACR | SLC2 | LY75 | SFRP1 | PTK2B |
| TP53 | HRX | MME | ACRB | SLCO1B1 | CBY1 | LEF1 | ELANE |
| BCR | HTRX1 | CD10 | CNGA1 | SLC22A8 | ARHGAP26 | DDIT3 | |
| WDSTS | CALLA | KCNMA1 | POLB | ST3GAL1 | GSTA1 | PTCH1 | |
| ABCB1 | CBL2 | NEP | CLCN2 | CDA | MIR199B | MECOM | CD247 |
| MTHFR | NSLL | CMT2T | IL17A | NT5E | ST8SIA4 | SRSF1 | STAT5B |
| TNF | CLLS5 | SCA43 | ADRB1 | DCTD | ATG4B | CDKN1C | AICDA |
| JAK2 | FLI1 | MLF1 | TUBB1 | ABCC10 | MIRLET7I | MIR17 | IDH2 |
| IL6 | BDPLT21 | LPP | CYP2E1 | SLC29A1 | PTBP2 | CRK | AXL |
| TGFB1 | ETV6 | CHIC2 | VDR | 1KBKG | SPRED2 | GATA2 | CDK9 |
| AKT1 | TEL | BTL | MPL | PRKCA | OSBP2 | NOTCH2 | PMP22 |
| GSTM1 | THC5 | PBT | CHRM1 | IMPDH1 | DDX43 | PRTN3 | ADIPOR1 |
| CTNNB1 | KRAS2 | RAP1GDS1 | CNRM2 | IMPDH2 | P2RX5 | IL32 | IKZF1 |
| KRAS | RASK2 | TCS1 | BCHE | PB1 | MKNK2 | MIR223 | TET2 |
| GSTT1 | NS | BST2 | UREC | NT5C2 | UBASH3B | IL24 | MTHFD1L |
| NFKB1 | CFC2 | DKCA2 | MMP12 | ENPP1 | MIR30E | ARRB1 | NFKB2 |
| BRCA1 | RALD | DKCB4 | NS5B | PRKCD | ATP5F1 | PAX5 | ERCC5 |
| MMP9 | CMTS | PFBMFT1 | ADRB2 | MS4A1 | KIR2DL5B | WSB1 | DAPK1 |
| STAT3 | PTPN11 | CMM9 | PTAFR | HCK | GAS2 | CIP2A | POU2F1 |
| ABL1 | PTP2C | LIFR | HRH1 | CDK2 | FAM27E5 | KIF11 | SPI1 |
| PTGS2 | SHP2 | SWS | NS5A | MAP2K1 | ETNK1 | MIR31 | SLC22A1 |
| CDKN2A | NS1 | STWS | ADRA2A | MAP2K2 | MIR1301 | BIN1 | SEP9 |
| IL1B | JMML | SJS2 | ADRA2B | MAP3K2 | ST8SIA6 | SET | |
| MYC | METCDS | ACSL6 | CHD1 | 1FNAR2 | LOC107126288 | JUP | |
| GSTP1 | CLLS2 | FACL6 | DRD2 | POLA1 | LOC107126281 | REL | |
| CXCL8 | D13S25 | ACS2 | DRD1 | SLC28A3 | MIR564 | HOXA9 | |
| LEP | DBM | IRF1 | HTR2A | PARP1 | MIR2278 | CRKL | |
| TERT | FLVCR2 | MAR | OPRM1 | PARP2 | MIR4701 | CSF3R | |
| BCL2 | C14orf58 | GRAF | PDE4B | PARP3 | ABL | SLCO1B3 | |
| IFNG | CCT | PDGFR | PANX1 | CD22 | GF1R | MTHFD1 | |
| MTOR | PVHH | IBGC4 | CYP3N4 | POLE | SPC | IFNAR1 | |
| XRCC1 | EPV | IMF1 | CASR | POLE2 | EPHA2 | EHMT2 | |
| FAS | SERPINA1 | PENTT | KCND | POLE3 | ICK | CDC6 | |
| CCND1 | PI | KOGS | HTR7 | POLE4 | YES1 | ADIPOR2 | |
| BIRC5 | AAT | NSD1 | ORM2 | PNP | KIT | PER3 | |
| GSK3B | TCL1B | ARA267 | SLC6A2 | C3 | FYN | KIR2DS2 | |
| MAPK14 | TML1 | STO | SMPD1 | C4A | BTK | EPHB4 | |
| ATM | TCL1A | SOTOS1 | HTR1A | C4B | NR4A3 | MEF2C | |
| MIR21 | TCL1 | CLLS4 | NOMO1 | C5 | CSK | ASXL1 | |
| HMGB1 | MYL | DEK | MAP2 | AOX1 | EPHA5 | HES1 | |
| CYP1A1 | CREBBP | D6S231E | PHD | DNMT1 | FGR | KIR2DL2 | |
| NOTCH1 | CBP | CTEPH1 | CA2 | SLC01A2 | FRK | PRAME | |
| KDR | RSTS1 | HLA-B | NR1I2 | HSD11B1 | HSPA8 | SMO | |
| NFE2L2 | MYH11 | SPDA1 | POMC | ALB | ZAK | ORM1 | |
| HLA-G | AAT4 | HLA-DPB1 | CALM1 | RARA | PPAT | MSR1 | |
| CASP3 | FAA4 | TREM2 | YARS | RARB | CYP3A4 | NUMB | |
| ABCG2 | FUS | MYB | TAT | 1KBKB | CYP1A2 | CAMK2G | |
| EZH2 | TLS | ALL2 | SLC16A2 | TXNRD1 | CYP1B1 | CCDC170 | |
| CDKN1B | ALS6 | MLSM7 | TFPI | MAPK3 | FM03 | GPX3 | |
| JUN | ETM4 | DEL7q | GNRHR | MAPK1 | RET | MIR451A | |
| ERCC2 | CBFB | C7DELq | KCNQ2 | CDKN1A | NTPK1 | CDK7 | |
| TNFSF10 | PEBP2B | NCF1 | KCNQ3 | HDAC1 | CSF1R | MIR101-1 | |
| RHOA | DIA4 | PRSS2 | HTR3A | PML | DDR1 | IRF8 | |
| WT1 | NMOR1 | TRY2 | GRIA1 | ADA | CYP3A7 | KIR2DS4 | |
| PDCD1 | CYBA | SCLL | GNB1 | CD38 | CYP2C9 | ID4 | |
| LGALS3 | NF1 | NSD3 | MRD42 | CD19 | CYP2D6 | CD33 | |
| CYP3A5 | VRNF | WHSC1L1 | CTRC | RXRA | CYP2C19 | KIR2DS1 | |
| CD274 | WSS | SLC20A2 | CLCR | RXRG | PTGS1 | HMMR | |
| KCNH2 | NFNS | MLVAR | IMD22 | 1GFBP3 | SLC22A2 | SOCS2 | |
| LCN2 | ERBB2 | GLVR2 | TPOR | PSG5 | ABCA3 | BLK | |
| AURKA | NGL | IBGC1 | MPLV | CSF2RA | CYP2C8 | RMND1 | |
| RUNX1 | NEU | NBN | THCYT2 | 1L3RA | UGT1A1 | MIR224 | |
| LEPR | HER2 | NBS1 | TAL1 | SDC2 | GSTA2 | RANGAP1 | |
| HSP90AA1 | MSF | THCYT3 | TCL5 | PRG2 | MGST2 | FUT1 | |
| NPM1 | MSF1 | LALL | SCL | EPOR | FLT3 | PCM1 | |
| AKAP12 | NAPB | BSAP | BCL10 | GPRC5A | RPI2 | MIR130A | |
| BCL2L1 | SH3GL1 | ALL3 | IMD37 | NROB1 | RPL3 | MIR7-1 | |
| MCL1 | EEN | TAL2 | GFI1 | ALDH1A2 | TEK | AHI1 | |
| IL2RA | LYL1 | CLLS3 | ZNF163 | RARRES1 | FGFR1 | CDKN2C | |
| PLK1 | CEBPA | CHDSKM | SCN2 | LCN1 | FGFR2 | ZBTB2 | |
| PTPN22 | CEBP | NUP214 | RBM15 | OBP2A | FGFR3 | PLCD1 | |
| XIAP | BCL3 | D9S46E | SPEN | RBP4 | FGFR4 | MTSS1 | |
| BCL2L11 | BAX | CAN | OTT | PDK4 | LCK | MSI2 | |
| DPP4 | TAM | CAIN | IGFR2 | CYP26A1 | SRC | FERMT3 | |
| SYK | MST | AF10 | CD32 | HPGDS | ABCB11 | PIWIL1 | |
| PDGFRA | CBFA2 | ALL1 | PBX1 | ATP1A1 | FCGR3B | RAPGEF1 | |
| MIR155 | AML1 | MBL2 | CAKUHED | DGUOK | C1R | MKNK1 | |
| TWIST1 | CML | MBL | ABL2 | 1TGAL | C1QA | EHMT1 | |
| CBL | PHL | MBP1 | ABLL | TOP2A | C1QB | USF2 | |
| STAT5A | ALL | MBL2D | ARG | PDLA1 | C1QC | MIR10A | |
| BMI1 | HMOX1 | MBPD | NCF2 | CBR1 | FCGR3A | IL1RAP | |
| HSPA4 | HMOX1D | LMO1 | FLVCR1 | AKR1A1 | C1S | MIR320A | |
| TGM2 | NCF4 | RBTN1 | AXPC1 | AKR1 | FCGR1A | LTB4R2 | |
| NFKBIA | P40PHOX | RHOM1 | PCARP | NQO1 | FCGR2A | SETBP1 | |
| CD34 | CGD3 | LMO2 | COPD | NOS3 | FCGR2B | ULBP2 | |
| CALR | MKL1 | RBTNL1 | TCL4 | NDUFS3 | FCGR2C | BTG1 | |
| MIR34A | AMKL | RHOM2 | ERBB4 | NDUFS7 | RRM2 | KDM5A | |
| XRCC3 | MAL | TTG2 | HER4 | POR | DCK | MLLT3 | |
| PDGFRB | XK | CLLS1 | ALS19 | ABCC3 | PRKAR2A | PHF6 | |
| SOCS1 | MCLDS | SMAR | SGOL1 | HPRT1 | PRKAR1A | CD7 | |
| ABCC1 | CYBB | NUMA1 | SGO | TUBB | PDE3A | PTPRG | |
| IFNA1 | CGD | PICALM | SGO1 | TUBA4A | 1FNAR1 | FCER1G | |
| PIK3CG | AMCBX2 | CALM | CAID | DHFR | FNTB | HULC | |
| CYP2B6 | IMD34 | CLTH | THRB | FPGS | PDGFD | MIR196B | |
| EIF4E | GATA1 | LAP | ERBA2 | TYMS | FLT1 | MR1 | |
| XPC | GF1 | ATA | THR1 | ATIC | FLT4 | RIN1 | |
| AURKB | ERYF1 | AT1 | PRTH | GGH | UGT1A3 | ST3GAL4 | |
| PTPN6 | NFE1 | ZBTB16 | MYD88 | FOLR1 | UGT1A4 | FIP1L1 | |
| DNMT3A | XLTDA | ZNF145 | MYD88D | IFNAR2 | UGT1A9 | MIR148B | |
| BCL6 | XLTT | PLZF | DCML | NS3 | UGT2B7 | MIR326 | |
| ALOX5 | XLANP | KMT2A | MONOMAC | 4A | UGT2B15 | MIR486-1 |