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. 2017 Dec 14;22(12):2221. doi: 10.3390/molecules22122221

Table 4.

Serotonergic GPCR panel of N-phenylsulfonyl indolines with different N′-substituents as measured in binding assays of four serotonin receptors (Ki values are in µM).

ID Structure 5-HT1A 5-HT2A 5-HT6 5-HT7
39a graphic file with name molecules-22-02221-i014.jpg not measured 4.76 0.76 55.76
39b graphic file with name molecules-22-02221-i015.jpg not active 26.85 6.60 not active
40a graphic file with name molecules-22-02221-i016.jpg not measured 4.52 1.85 40.17
40b graphic file with name molecules-22-02221-i017.jpg not measured 3.82 2.42 not active