Table 1.
Compound | EC50 (µM) | ||
---|---|---|---|
A549 | MCF-7 | U87 | |
1 | 19.6 ± 4.5 | 21.6 ± 3.6 | 15.5 ± 5.4 |
2 | >100.0 | >100.0 | >100.0 |
3 | 36.3 ± 4.6 | 12.6 ± 2.6 | 14.2 ± 4.8 |
4 | >100.0 | >100.0 | >100.0 |
5 | 19.8 ± 8.3 | 36.0 ± 0.3 | 72.6 ± 4.6 |
6 | 75.3 ± 5.7 | 69.3 ± 3.5 | 80.4 ± 6.8 |
7 | 6.8 ± 0.6 | 11.2 ± 1.1 | 30.8 ± 2.8 |
8 | >100.0 | 30.0 ± 0.6 | 59.8 ± 8.7 |
9 | 22.1 ± 2.0 | 16.2 ± 4.2 | >100.0 |
10 | 37.6 ± 2.7 | 19.0 ± 5.7 | 59.5 ± 3.8 |
11 | 69.2 ± 0.6 | 23.1 ± 5.5 | 88.4 ± 14.4 |
12 | >100.0 | >100.0 | >100.0 |
13 | >100.0 | 15.9 ± 4.3 | >100.0 |
14 | >100.0 | >100.0 | >100.0 |
15 | >100.0 | 71.5 ± 13.6 | 73.8 ± 13.6 |
API | 77.5 ± 9.2 | 71.5 ± 15.6 | >100.0 |
BCL | 68.2 ± 3.6 | 26.1 ± 7.1 | >100.0 |