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Enzyme inhibition values for the INH derivatives. Results are expressed as a percentage of InhA inhibition.
| Compound | % Inhibition at 50 μM (Inhibitor) | Compound | % Inhibition at 50 μM (Inhibitor) |
|---|---|---|---|
| 1a | 45 | 5 | 19 |
| 1b | 54 | 6 | 43 |
| 1c | 48 | 7 | 39 |
| 1d | 64 | 8 | 42 |
| 2 | 54 | 9 | 32 |
| 3 | 3 | 10 | 79 |
| 4 | 33 | 11 | not soluble |
| TCL | >99 |
