Table 4.
Inhibitory activity of 3d and its analogs (10 nM) on histamine release in RBL-2H3 cells.
Compound | % Inhibition |
---|---|
3d | 53 |
6a | 52 |
6b | 48 |
6c | 32 |
6d | 18 |
6e | 55 |
6f | −42 |
6g | 4 |
6h | −26 |
6i | 11 |
Inhibitory activity of 3d and its analogs (10 nM) on histamine release in RBL-2H3 cells.
Compound | % Inhibition |
---|---|
3d | 53 |
6a | 52 |
6b | 48 |
6c | 32 |
6d | 18 |
6e | 55 |
6f | −42 |
6g | 4 |
6h | −26 |
6i | 11 |