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. Author manuscript; available in PMC: 2019 Sep 1.
Published in final edited form as: Bioorg Med Chem Lett. 2018 Apr 7;28(16):2697–2700. doi: 10.1016/j.bmcl.2018.04.003

Figure 2.

Figure 2

Preparation of β-hydroxy difluoromethyl ketones 49 and β-amino difluoromethyl ketones 1014. Isolated yields for the aldol and imino-aldol reactions are given in parenthesis.