Table 4.
The thio-functionalized carbohydrate derivatives used in this study.
| Compound | LogP/cLog | References |
|---|---|---|
| 5-thio-D-glucose pentaacetate (1) | LogP: −0.51 cLog: 0.72825 |
[19] |
| 6-thio-β-d-fructopyranose (2) | LogP: −1.36 cLog: −1.9984 |
[19] |
| 1,6-anhydro-5-C-hydroxymethyl-α-l-altro-pyranose (3) | LogP: −2.38 cLog: −1.5973 |
[19] |
| 2-C-methylene-myo-inositol oxide (4) | LogP: −3.22 cLog: −11214 |
[19] |
| 1,5-anhydro-6-deoxy-6-methanesulfamido-d-glucitol (5) | LogP: −3.6 cLog: −1.1515 |
[19] |
| 1,6-anhydro-3-deoxy-4-S-(2,3,4,6-tetra-O-acetyl-β-d-glucopyranosyl-d-glycero-hexopyranos-2-ulose (6) | LogP: −1.13 cLog: 0.4407 |
[18,42] |
| 1,6-anhydro-3-deoxy-4-S-β-d-glucopyranosyl-d-glycero-hexopyranos-2-ulose (7) | LogP: −2.05 cLog: −1.69975 |
[18,42] |
| 1,6-anhydro-3-deoxy-4-S-β-salicylyl-d-glycero-hexopyranos-2-ulose (8) | LogP: 1.28 cLog: 0.8949 |
[43] |
| 1,6-anhydro-3-deoxy-4-S-(2,3,4,6-tetra-O-acetyl-β-d-galactopyranosyl-d-glycero-hexopyranos-2-ulose (9) | LogP: −1.13 cLog: 0.4407 |
[18,42] |
| 2-acetamido-2-dexy-1,5-anhydro-d-mannitol (10) | Log P: −2.75 cLog: 0.993001 |
[44] |
| 1,2-O-isopropylidene-5,6-anhydro-3-hydroxy-d-glucofuranose (11) | LogP: −0.39 cLog: 0.64599 |
[45] |
| 1,2-O-isopropylidene-3,5-di-O-acetyl-6-methoxy-d-glucofuranose (12) | LogP: −0.2 cLog: 0.9672 |
[46] |
| 1-C-nitromethyl-d-gluco-pyranose (13) | LogP: −4.22 cLog: −1.9428 |
[47] |
| 1,6-anhydro-3,4-dideoxy-α-d-glycero-hex-3-enopyranos-2-thiosemicarbazone (14) | LogP:−0.18 cLog:0.372 |
[48,49] |
| 1,6-anhydro-3-deoxy-4-S-(octa-O-acetyl-β-d-lactosyl-d-glycero-hexopyranos-2-ulose (16) | LogP:−2.18 cLog:0.854498 |
[48,49] |
| 1,6-anhydro-3,4-dideoxy-α-d-glycero-hexopyranos-2-thiosemicarbazone (14A) | LogP: −0.29 cLog: 0.204 |
[48,49] |
| 1,6-anhydro-3-deoxy-4-S-(octa-O-acetyl-β-d-lactosyl-d-glycero-hexopyranos-2-thiosemicarbazone (16A) | LogP: NA cLog: 1.26 |
[48,49] |
| Octa-O-acetyl-β-d-lactosyl-S-1-adamantane (19) | cLog: 4.0538 | [49] |
| 1,6-anhydro-3-deoxy-4-S-(2,3,4-tri-O-acetyl-β-l-arabino)-d-glycero-hexopyranos-2-ulose (20) | LogP: −0.9 cLog: 0.632201 |
[49] |
| 1,6-anhydro-3-deoxy-4-S-(5-amino-1,3,4-thiadiazol-2-yl)-d-glycero-hexopyranos-2-ulose (23) | LogP: 1.37 cLog: −0.535599 |
[50] & this work |
| 1,6-anhydro-3-deoxy-4-S-(4,5-dihydrothiazol-2-yl-d-glycero-hexopyranos-2-ulose (26) | LogP: 1.13 cLog: 0.0390999 |
[50] & this work |