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. Author manuscript; available in PMC: 2019 Jun 30.
Published in final edited form as: Tetrahedron. 2018 Jul 17;74(35):4592–4600. doi: 10.1016/j.tet.2018.07.027

Table 2.

Synthesized drug-like library of acetylated imidazo[1,2-a]pyridines.

Compd Structure Yielda (%) Compd Structure Yielda (%)
9 graphic file with name nihms-987520-t0002.jpg 99 20 graphic file with name nihms-987520-t0003.jpg 85
10 graphic file with name nihms-987520-t0004.jpg 62 21 graphic file with name nihms-987520-t0005.jpg 90
11 graphic file with name nihms-987520-t0006.jpg 92 22 graphic file with name nihms-987520-t0007.jpg 54
12 graphic file with name nihms-987520-t0008.jpg 83 23 graphic file with name nihms-987520-t0009.jpg 50
13 graphic file with name nihms-987520-t0010.jpg 99 24 graphic file with name nihms-987520-t0011.jpg 55
14 graphic file with name nihms-987520-t0012.jpg 85 25 graphic file with name nihms-987520-t0013.jpg 73
15 graphic file with name nihms-987520-t0014.jpg 81 26 graphic file with name nihms-987520-t0015.jpg 81
16 graphic file with name nihms-987520-t0016.jpg 70 27 graphic file with name nihms-987520-t0017.jpg 84
17 graphic file with name nihms-987520-t0018.jpg 99 28 graphic file with name nihms-987520-t0019.jpg 95
18 graphic file with name nihms-987520-t0020.jpg 74 29 graphic file with name nihms-987520-t0021.jpg 76
19 graphic file with name nihms-987520-t0022.jpg 79 30 graphic file with name nihms-987520-t0023.jpg 53
31 graphic file with name nihms-987520-t0024.jpg 56 42 graphic file with name nihms-987520-t0025.jpg 83
32 graphic file with name nihms-987520-t0026.jpg 70 43 graphic file with name nihms-987520-t0027.jpg 62
33 graphic file with name nihms-987520-t0028.jpg 71 44 graphic file with name nihms-987520-t0029.jpg 80
34 graphic file with name nihms-987520-t0030.jpg 50 45 graphic file with name nihms-987520-t0031.jpg 75
35 graphic file with name nihms-987520-t0032.jpg 73 46 graphic file with name nihms-987520-t0033.jpg 20
36 graphic file with name nihms-987520-t0034.jpg 60
37 graphic file with name nihms-987520-t0035.jpg 45b
38 graphic file with name nihms-987520-t0036.jpg 75
39 graphic file with name nihms-987520-t0037.jpg 87
40 graphic file with name nihms-987520-t0038.jpg 85
41 graphic file with name nihms-987520-t0039.jpg 60
a

Isolated Yield.

b

Continued for 24 h.