Table 6.
Receptor | Hot Ligand | Hot Ligand Activity | (±)-MDMA | R-(−)-MDMA | S-(+)-MDMA |
---|---|---|---|---|---|
5-HT 1 | 3H-5-HT | Agonist | 6,850 ± 1,300 | 4,200 ± 500 | >10,000 |
5-HT2 | 3H-Ketanserin | Antagonist | 8,300 ± 1,100 | 3,310 ± 140 | >10,000 |
D2 | 3H-NMSP | Antagonist | >10,000 | >10,000 | >10,000 |