(a,d) Representative traces of mEPSCs recorded from control
rat hippocampal neurons or neurons with cypin knockdown treated with vehicle
(<0.1% DMSO; control; n=17/23) or 20 μM of the following
compounds: H9, (n=6/8), B9 (n=7/8), G5 (n=13/11), or G6 (n=9/8). n=number of
neurons/number of cultures. (b,c,e,f) Bar graph analysis of mEPSC
frequency and amplitude following 48 hour baseline drug treatment. Pretreatment
with H9 increases the frequency of mEPSCs in control neurons with no change to
amplitude. (g,j) Representative traces of mEPSCs recorded from rat
hippocampal neurons treated with vehicle (<0.1% DMSO; control; n=17/23),
or 20μM of the following compounds: NMDA (n=19/16), H9 + NMDA (n=12/12),
B9 + NMDA (n=15/11), G5 + NMDA (n=17/12), and G6 + NMDA (n=12/8). n=number of
neurons/number of cultures. (h,i,k,l) Bar graph analysis of mEPSC
frequency and amplitude following 48 hour drug treatment, 5 minute 20 μM
NMDA-induced injury, and two hour recovery period. Treatment with cypin
activators prevents the decrease in frequency and amplitude induced by NMDA
injury in control neurons, while cypin knockdown causes a loss of function and
subsequent decrease of mEPSC frequency and amplitude.
*p<0.05, **p<0.01,
***p<0.005, ****p<0.001
determined by one-way ANOVA followed by Tukey-Kramer multiple comparisons test.
Error bars indicate mean ± SEM.