Table 1.

In vitro activity of the hits identified by WHALES-GM on RXRα/β/γ. EC₅₀ ± SEM [µM] is reported (n ≥ 4).

ID	Compound	RXRα [µM]	RXRβ [µM]	RXRγ [µM]
5		17 ± 1	14.7 ± 0.8	15.0 ± 0.6
6		16.5 ± 0.6	16.6 ± 0.2	16 ± 4
7		32.1 ± 0.9	25.1 ± 0.1	28.2 ± 0.1
8		23.7 ± 0.7	25.6 ± 0.4	32 ± 3