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. 2018 Sep 17;23(9):2369. doi: 10.3390/molecules23092369
ABCB1 ATP-binding cassette sub-family B member 1
ALL acute lymphoblastic leukemia
Bcr-Abl breakpoint cluster region-Abelson
Btk Bruton’s tyrosine kinase
CML chronic myeloid leukemia
c-Src cellular-sarcoma tyrosine kinase
DIPEA N,N-diisopropylethylamine
EMA European Medicines Agency
FDA Food and Drug Admnistration
FRET fluorescence resonance energy transfer
GBM glioblastoma multiforme
HRI hydrophobic region I
HTS high-throughput screening
NB neuroblastoma
NCEs new chemical entities
PDGFR platelet derived growth factor receptor
Ph+ Philadelphia chromosome–positive
RET REarranged during Transfection
SFK Src family kinase
SH Src homology
STK serine/threonine kinase
TK tyrosine kinase
VEGFR vascular endothelial growth factor