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. Author manuscript; available in PMC: 2019 Nov 21.
Published in final edited form as: J Med Chem. 2018 Nov 8;61(22):10299–10309. doi: 10.1021/acs.jmedchem.8b01487

Scheme 1.

Scheme 1.

Synthesis of RTS-V5.a

a Reagents and conditions: a) HATU, DIPEA, DMF, rt, 16 h. b) TFA, CH2Cl2, rt, 4 h. c) 4-((Benzyloxy)carbamoyl)benzoic acid, HATU, DIPEA, DMF, rt, 24 h. d) Pd/C, H2, rt, 4 h.