Table 2.
Entry | 2-Aminoaryl ketone | CH-acid | Product | Yield (%)a | Mp (˚C) Found | Mp (˚C) Reported |
1 | 90 | 102-103 | 100-101b | |||
2 | 92 | 110-112 | 111-112b | |||
3 | 94 | 153-154 | 156-157c | |||
4 | 90 | 130-131 | 130-132c | |||
5 | 89 | 192-194 | 190-192c | |||
6 | 92 | 155-157 | 155-156c | |||
7 | 93 | 99-100 | 98-100d | |||
8 | 95 | 152-154 | 153-154e | |||
9 | 94 | 103-105 | 105-107f | |||
10 | 95 | 164-166 | 164-165c | |||
11 | 91 | 150-152 | 150-151c | |||
12 | 89 | 186-187 | 185-186c | |||
13 | 88 | 106-108 | 106-107b | |||
14 | 92 | 207-209 | 208-209c | |||
15 | 94 | 132-134 | 133-135b |