Table 8.
HDAC inhibitors with effects on non-coding RNA tumor suppressors (inducing effects) and oncogenes (suppressing effects) in mesothelioma correlated with gemcitabine or pemetrexed activity.
Drugs | Tumor suppressors | Oncogenes |
---|---|---|
NaB | miR-15/16, miR-126, miR-202, miR-143, miR-145 | – |
NaPBA | miR-34a, miR-148a | – |
TSA | let-7b, let-7c, miR-15/16, miR-34a, miR-126, miR-202, miR-203, miR-486 | – |
SAHA | let-7d, miR-15a, miR-16, miR-34b | HOTAIR |
AR-42 | let-7b, let-7d, miR-15b, miR-34a | miR-17-5p, miR-21 |
LAQ824 | – | miR-21 |
Panobinostat | let-7b, miR-15a, miR-16 | – |