Table 2.
Entry | Aryl- | Product | Yield % |
---|---|---|---|
1 | Ph- | 7f | 85 |
2 | 4-F-Ph- | 7g | 71 |
3 | 2-Tolyl- | 7 h | 65 |
Reaction conditions: arylboronic acid (4 equiv.), Pd(PPh3)4 (2.5 mol %), Na2CO3 (4 equiv.), DME/ethanol (9:1), MW 300 W, 80 °C, 3 h
Entry | Aryl- | Product | Yield % |
---|---|---|---|
1 | Ph- | 7f | 85 |
2 | 4-F-Ph- | 7g | 71 |
3 | 2-Tolyl- | 7 h | 65 |
Reaction conditions: arylboronic acid (4 equiv.), Pd(PPh3)4 (2.5 mol %), Na2CO3 (4 equiv.), DME/ethanol (9:1), MW 300 W, 80 °C, 3 h