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Inhibition of the compounds for the relatively receptor.
| Compound | Concentration (mol/L) | Emax10 μM a (%) | |||||
|---|---|---|---|---|---|---|---|
| μ | δ | κ | 5-HT2A | 5-HT1A | 5-HT uptake | ||
| Naloxone | 10-5 | 100 | 100 | 100 | - | - | - |
| Aripiprazole | 10-5 | - | - | - | 100 | - | - |
| 5-HT | 10-5 | - | - | - | - | 100 | - |
| Duloxetine | 10-5 | - | - | - | - | - | 90.6 |
| w-conotoxinGVIA | 10-5 | - | - | - | - | - | - |
| 18 | 10-5 | 18.1 | 0 | 2.9 | 57.7 | 96.9 | 59.3 |
a Maximal inhibition effect at the highest tested concentration (Emax10 μM).
