Table 3.
Library | Rank | ZINC ID | Structure | Binding Energy (kcal/mol) | xlogP | H-bond Donors | H-bond Acceptors | Molecular Weight (g/mol) |
---|---|---|---|---|---|---|---|---|
Ref | R | ZINC03817234 | −10.2 | −3.50 | 2 | 6 | 514.69 | |
S * | 1 | ZINC71849549 | −12.2 | 2.27 | 2 | 6 | 318.89 | |
P ** | 2 | ZINC00825224 | −12.0 | 4.11 | 3 | 5 | 397.488 | |
P | 3 | ZINC00634884 | −12.0 | 5.96 | 1 | 6 | 481.60 | |
S | 4 | ZINC32760563 | −11.9 | 3.47 | 0 | 5 | 388.51 | |
S | 5 | ZINC32760533 | −11.8 | 3.44 | 0 | 5 | 388.52 | |
S | 6 | ZINC25010434 | −11.8 | 2.16 | 1 | 7 | 431.54 | |
P | 7 | ZINC00851466 | −11.8 | 5.52 | 3 | 10 | 536.38 | |
S | 8 | ZINC71818945 | −11.7 | 3.35 | 0 | 6 | 434.58 | |
P | 9 | ZINC00895646 | −11.7 | 3.99 | 2 | 7 | 451.55 | |
P | 10 | ZINC00895634 | −11.7 | 3.54 | 2 | 7 | 438.53 |
* Similarity-based library, ** Pharmacophore-based library, Ref-Maraviroc.