Table 5.
-R1 | -R2 | Compound | Time a (h) | Yield b (%) |
---|---|---|---|---|
H | 14a | 0.5 | 80 | |
H | 14b | 0.5 | 96 | |
H | 14c | 0.5 | 89 | |
H | 14d | 0.5 | 88 | |
14e | 0.5 | 87 | ||
14f | 0.5 | 86 |
a Time of the conversion of 13 into the corresponding thioureas (step 1); b Isolated yield.
-R1 | -R2 | Compound | Time a (h) | Yield b (%) |
---|---|---|---|---|
H | 14a | 0.5 | 80 | |
H | 14b | 0.5 | 96 | |
H | 14c | 0.5 | 89 | |
H | 14d | 0.5 | 88 | |
14e | 0.5 | 87 | ||
14f | 0.5 | 86 |
a Time of the conversion of 13 into the corresponding thioureas (step 1); b Isolated yield.